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Referencia número: HY-175306

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GPR183 inverse agonist-1

GPR183 inverse agonist-1 (Compound 78) is a GPR183 inverse agonist. GPR183 inverse agonist-1 inhibits the GPR183-mediated Gi activation and β-arrestin2 recruitment, and blocks PBMC migration. GPR183 inverse agonist-1 can be used for inflammatory, autoimmune and neoplastic disorders research.

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No. CAS: 2380033-51-0
Fòrmula: C₂₀H₂₀BrN₅O₂
Peso molecular:442.31

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Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (267 KB)

GPR183 inverse agonist-1 Chemical Structure

No. CAS: 2380033-51-0

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IC₅₀ & Target^[1]

Arrestin-3/β-Arrestin 2

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Chemical Information

No. CAS 2380033-51-0
Peso molecular 442.31
Fòrmula C₂₀H₂₀BrN₅O₂
SMILES

O=C(C1=CC=C(Br)C=C1)N(CC2)CCC2CN3C(C=CC(N4N=CC=C4)=N3)=O
Envío

Room temperature in continental US; may vary elsewhere.
Almacenamiento

Please store the product under the recommended conditions in the Certificate of Analysis.

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Pureza: 99.98%

Assay: 99.98%

ee.: 99.98%

Ficha de datos (267 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Instrucciones de manejo (2659 KB)

Referencias

[1]. Andersson L, et al. AI-Driven Virtual Screening and First-in-Class Conformational Biosensor Enable the Discovery of a GPR183 Inverse Agonist[J]. bioRxiv, 2025: 2025.06. 19.659764.

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How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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GPR183 inverse agonist-1

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GPR183 inverse agonist-1

Ver todos los productos específicos de isoformas Arrestin

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GPR183 inverse agonist-1 Related Classifications

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