hCAIX-IN-21
hCAIX-IN-21 (compound 16c) is a potent hCAIX inhibitor with KI values of 5.2, 3.5, 12.6, 13600 nM for hCAIX, hCA II, hCA XII, hCA I, respectively. hCAIX-IN-21 inhibits cathepsin B enzyme activity.
For research use only. We do not sell to patients.
- CAS No.: 3047757-55-8
- Formula: C20H17FN6O4S
- Molecular Weight:456.45
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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hCA IX 5.2 nM (Ki) |
hCA II 3.5 nM (Ki) |
hCA XII 12.6 nM (Ki) |
hCA I 13600 nM (Ki) |
Chemical Information
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CAS No. 3047757-55-8
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Molecular Weight 456.45
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Formula C20H17FN6O4S
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SMILES
O=C(C1=NN(C2=CC=C(S(=O)(N)=O)C=C2)C(C3=C(C)N(C4=CC=C(F)C=C4)N=N3)=C1)OC
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)