S9-CMC1 TFA
S9-CMC1 TFA is a covalent peptide lysine-specific demethylase 1 (LSD1) inhibitor with an IC50 value of 2.53 μM. S9-CMC1 TFA specifically recognizes Cys360 in the enzyme-active region. S9-CMC1 TFA inhibits LSD1 activity, increasing H3K4me1 and H3K4me2 levels, leading to G1 cell cycle arrest and apoptosis and inhibiting cell proliferation. S9-CMC1 TFA significantly inhibits tumor growth in A549 xenograft animal models.
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- 화학식: C97H151F3N32O17S2
- 분자량:2158.57
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보관:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- 순도&문서
- References
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Help & FAQs
Biological Activity
Chemical Information
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분자량 2158.57
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화학식 C97H151F3N32O17S2
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Sequence
Ac-Pro-Arg-cyclo(Cys-Phe-Leu-Val-Met)-Lys-Pro-Arg-Arg-Arg-Arg-Trp-NH2 (Cyclization Bridge via Benzene-1,3-bismethylene: Cys3-Met7)
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Sequence Shortening
Ac-PR-Cyclo(CFLVM)-KPRRRRW-NH2 (Cyclization Bridge via Benzene-1,3-bismethylene: Cys3-Met7)
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선적
Room temperature in continental US; may vary elsewhere.
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보관
Please store the product under the recommended conditions in the Certificate of Analysis.
순도&문서
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
S9-CMC1 TFA Related Classifications
HY-P10819 Related Classifications
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