MOR agonist-2
MOR agonist-2 (compound 46) is a antagonist of D3R and agonist of MOR (Ki: 7.26 nM and 564 nM, respectively). MOR agonist-2 has the potential to produce analgesic effects through MOR partial agonism. MOR agonist-2 reduces opioid-misuse liability via D3R antagonism.
For research use only. We do not sell to patients.
- CAS No.: 2833692-02-5
- Formula: C37H47Cl2N5O3
- Molecular Weight:680.71
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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D3 Receptor |
μ Opioid Receptor/MOR |
Chemical Information
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CAS No. 2833692-02-5
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Molecular Weight 680.71
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Formula C37H47Cl2N5O3
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SMILES
O=C([C@H]1N(CCC(C2=CC=CC=C2)(C3=CC=CC=C3)C(N(C)C)=O)C[C@H](O)C1)NCCCCN4CCN(C5=CC=CC(Cl)=C5Cl)CC4
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)