Naldemedine

(Synonyms: S-297995)
2 Cited Publications
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Based on 2 publication(s) in Google Scholar

Naldemedine (S-297995) is an orally active μ-opioid receptor antagonist (PAMORA). Naldemedine shows potent binding affinities (Ki=0.34, 0.43, 0.94 nM, respectively) and antagonist activities (IC50=25.57, 7.09, 16.1 nM, respectively) for recombinant human μ-, δ-, and κ- opioid receptors. Naldemedine can be used in opioid-induced constipation (OIC) research. Naldemedine is predicted to bind to 3CLpro encoded by SARS-CoV2 genome.

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  • CAS No.: 916072-89-4
  • Formule: C32H34N4O6
  • Masse moléculaire:570.64
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    Please store the product under the recommended conditions in the Certificate of Analysis.

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