PG-911
PG-911 is a full MC5R agonist (EC50 = 0.031 nM for hMC5R). PG-911 is also a full antagonist at the hMC3R and the hMC4R (Kb: 0.38 nM and 0.17 nM, respectively). PG-911 can be used in the research of neurological disorders.
For research use only. We do not sell to patients.
- Formula: C53H71N13O10
- Molecular Weight:1050.21
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
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hMC5R 0.031 nM (EC50) |
hMC3R 0.38 nM (Kb) |
hMC4R 0.17 nM (Kb) |
Chemical Information
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Molecular Weight 1050.21
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Formula C53H71N13O10
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Sequence
Ac-{Nle}-cyclo(Asp-{Hyp}-{d-Nal}-Arg-Trp-Lys)
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Sequence Shortening
Ac-{Nle}-cyclo(D-{Hyp}-{d-Nal}-RWK)
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
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