PAK1-IN-2
PAK1-IN-2 (Compound 35) is a selective PAK1 inhibitor with a Ki of 7.3 nM. PAK1-IN-2 can inhibit MEK phosphorylation. PAK1-IN-2 has significant inhibitory effects on PAK1/4 amplified cancer cell lines. PAK1-IN-2 can be used in the study of cancer.
For research use only. We do not sell to patients.
- Formula: C21H24N8OS
- Molecular Weight:436.53
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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PAK1 7.3 nM (Ki) |
Chemical Information
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Molecular Weight 436.53
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Formula C21H24N8OS
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SMILES
CN(C(C1(C#N)CNC1)=O)C2(C3)CC3(C2)NC4=NC(NC5=NC=C(C6CC6)S5)=CC=N4
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)