PCAF/GCN5 ligand 1
PCAF/GCN5 ligand 1 is a PCAF/GCN5 ligand with high binding affinity. PCAF/GCN5 ligand 1 shows no functional effect on PCAF/GCN5 activity. PCAF/GCN5 ligand 1 undergoes optimization into a potent and selective PCAF/GCN5 ligand GSK4027 (HY-101027).
For research use only. We do not sell to patients.
- CAS No.: 1209224-91-8
- Formula: C12H11ClFN3O
- Molecular Weight:267.69
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
PCAF/GCN5 ligand 1 (Compound 8) (10 μM) binds to the purified PCAF bromodomain with low micromolar affinity and good ligand efficiency[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 1209224-91-8
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Molecular Weight 267.69
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Formula C12H11ClFN3O
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SMILES
CN1N=CC(NCC2=CC=C(F)C=C2)=C(Cl)C1=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
PCAF/GCN5 ligand 1 Related Classifications
HY-181279 Related Classifications
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