PF 02367982
PF 02367982 is a potent and select progesterone receptor (PR) antagonist with an IC50 value of 47.3 nM. PF 02367982 has oral activity.
For research use only. We do not sell to patients.
- CAS No.: 913344-84-0
- Formula: C19H20N4O2
- Molecular Weight:336.39
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
Chemical Information
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CAS No. 913344-84-0
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Molecular Weight 336.39
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Formula C19H20N4O2
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SMILES
O=C(NC)CN1N=C(C2CC2)C(OC3=CC=C(C#N)C=C3)=C1C4CC4
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
[1]. Alexander de Giorgio-Miller, et al. The translational pharmacology of a novel, potent, and selective nonsteroidal progesterone receptor antagonist, 2-[4-(4-cyano-phenoxy)-3,5-dicyclopropyl-1H-pyrazol-1-yl]-N-methylacetamide (PF-02367982). J Pharmacol Exp Ther. 2008 Oct;327(1):78-87. [Content Brief]
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)