Scientific Reviews
Product Guides
Blogs
Topics
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
79 Results for "
Inactive metabolite
" in MedChemExpress (MCE) Product Catalog:
Products (79)
79 Results for "Inactive metabolite" in MCE Product Catalog:
Cat. No.: HY-W759719
Synonyms: 21-desDFZ-d4
Cat. No.: HY-W704807
CAS No.: 2409015-09-2
Synonyms: 3-O-methyl Dopamine-d3 hydrochloride
Cat. No.: HY-W745860
CAS No.: 2469279-20-5
Target:
Research Areas:
13,14-Dihydro-15-keto-PGE1 is an inactive metabolite of PGE1. 13, 14-Dihydro-15-Keto-pGE1 inhibited platelet aggregation in ADP-induced human isolated platelet-rich plasma with IC50 14.8 μg/mL .
Cat. No.: HY-134520R
CAS No.: 13649-88-2
Research Areas:
21-Deacetoxy deflazacort (Standard) is the analytical standard of 21-Deacetoxy deflazacort. This product is intended for research and analytical applications. 21-Deacetoxy deflazacort is a dehydrogenated derivative of Deflazacort (HY-13609), a glucocorticoid, an inactive precursor that is rapidly converted to the active metabolite 21-Desacetyldeflazacort. Deflazacort acts as an anti-inflammatory and immunosuppressant .
Cat. No.: HY-137551R
CAS No.: 1220411-29-9
Target:
Research Areas:
21-Deacetoxy deflazacort (Standard) is the analytical standard of 21-Deacetoxy deflazacort. This product is intended for research and analytical applications. 21-Deacetoxy deflazacort is a dehydrogenated derivative of Deflazacort (HY-13609), a glucocorticoid, an inactive precursor that is rapidly converted to the active metabolite 21-Desacetyldeflazacort. Deflazacort acts as an anti-inflammatory and immunosuppressant .
Cat. No.: HY-113083R
CAS No.: 16110-10-4
Synonyms: APAP-glu (Standard)
Category:
Cat. No.: HY-W653919
Cat. No.: HY-W014109
CAS No.: 69304-49-0
Synonyms: (E)-5-(2-Bromovinyl)uracil; BVU
Target:
Research Areas:
(E)-5-(2-Bromovinyl)uracil (BVU) is a pyrimidine base and an inactive metabolite of the antiviral agents sorivudine and (E)-5-(2-bromovinyl)-2'-deoxyuridine (BVDU) that may be regenerated to BVDU in vivo. BVU irreversibly inactivates dihydropyrimidine dehydrogenase (DPD) in an NADPH-dependent manner. It enhances the efficacy of the chemotherapeutic agent and DPD substrate 5-fluorouracil (HY-90006) in a P388 murine leukemia model when administered at a dose of 200 μmol/kg, increasing survival time.
Cat. No.: HY-126194
CAS No.: 204853-33-8
Synonyms: Ro 61-1448
Cat. No.: HY-136913R
CAS No.: 69617-84-1
Synonyms: (Rac)-Betuligenol (Standard)
Research Areas:
(Rac)-Rhododendrol (Standard) ((Rac)-Betuligenol (Standard)) is the analytical standard of (Rac)-Rhododendrol (HY-136913). This product is intended for research and analytical applications. (Rac)-Rhododendrol ((Rac)-Betuligenol) is an aromatic compound with pro-oxidant activity. (Rac)-Rhododendrol may be useful in the suppression of liver diseases. (Rac)-Rhododendrol can be toxic to melanocytes, leading to cell death. The metabolite of (Rac)-Rhododendrol, RD-quinone, is cytotoxic and causes enzyme inactivation and endoplasmic reticulum stress by binding to thiol proteins. (Rac)-Rhododendrol-derived melanin exhibits potent pro-oxidant activity and may cause oxidative stress .
Cat. No.: HY-W738271
CAS No.: 91384-88-2
Synonyms: 3,4-Dimethoxybenzyl alcohol-13C
Category:
Cat. No.: HY-127025
CAS No.: 61443-77-4
Target:
Research Areas:
8-Hydroxy loxapine is the relatively inactive oxidative metabolite of Loxapine (HY-17390), compared to 7-OH-loxapine .
Cat. No.: HY-113083A
Synonyms: APAP-glu potassium
Target:
Research Areas:
Acetaminophen glucuronide potassium (APAP-glu potassium) is the inactive glucuronide metabolite of Acetaminophen (HY-66005). Acetaminophen glucuronide potassium can be used as a biomarker to measure glucuronidation activity or hepatic drug metabolism capacity .
Cat. No.: HY-127025S1
Cat. No.: HY-126373S
Synonyms: SN-38G-d5
Cat. No.: HY-182445
CAS No.: 140369-78-4
Research Areas:
FPL 66564 is a short-acting angiotensin-converting enzyme (ACE) inhibitor with an IC50 of 5.7 nM against rabbit ACE. FPL 66564 inhibits ACE activity at the functional level and is hydrolyzed in human blood into inactive hydrophilic metabolites. FPL 66564 modulates angiotensin I-induced pressor responses in anesthetized rats, and its effects rapidly return to baseline after cessation of intravenous infusion. FPL 66564 can be used for research on cardiovascular regulation related to critical illness .
-
-
Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
