6 Results for "

NTS2

" in MedChemExpress (MCE) Product Catalog:
Products (6)

6 Results for "NTS2" in MCE Product Catalog:

Cat. No.: HY-P2544
CAS No.: 139026-64-5
Synonyms: JMV438
Target:  

Neurotensin Receptor

Research Areas:  

Neurological Disease

[Lys8, Lys9]-Neurotensin (8-13) (JMV438), a Neurotensin analog, exerts its analgesic effects through activation of the G protein-coupled receptors NTS1 and NTS2, with Ki values of 0.33 nM and 0.95 nM for hNTS1 and hNTS2 receptors, respectively .
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Cat. No.: HY-12436
CAS No.: 1623002-61-8
Purity:  98.2%
Target:  

Neurotensin Receptor

Research Areas:  

Neurological Disease

NTRC-824 (Compound 5) is a potent, selective and neurotensin-like nonpeptide neurotensin receptor type 2 (NTS2) antagonist with an IC50 of 38 nM and a Ki of 202 nM. NTRC-824 is >150-fold selectivity for NTS2 over NTS1 (Ki >30 μM) .
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Cat. No.: HY-124831
CAS No.: 1811503-67-9
Target:  

Neurotensin Receptor

Research Areas:  

Neurological Disease

NTRC-844 (compound 8) is a selective antagonist of neurotensin receptor type 2 (NTS2),with the EC50 of 238 nM. NTRC-844 plays an important role in analgesic animal research .
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Cat. No.: HY-137525
CAS No.: 1643879-88-2
Target:  

Neurotensin Receptor

Research Areas:  

Neurological Disease

NTRC-808 is a nonpeptide selective GPCR neurotensin receptor type 2 (NTS2) partial agonist with an EC50 of 14 nM and Ki of 88 nM. NTRC-808 has higher selectivity for NTS2 than for NTS1. NTRC-808 has antipsychotic and analgesic activity .
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Cat. No.: HY-P10767
CAS No.: 2468971-42-6
Target:  

Neurotensin Receptor

Research Areas:  

Neurological Disease

MD01-67 is a selective macrocyclic compound targeting the neurotensin receptor type 2 (NTS2), with Ki of 2.9 nM. MD01-67 exhibits analgesic and tactile hypersensitivity reducing activity in rats acute/persistent/chronic inflammatory pain models .
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Cat. No.: HY-12217
CAS No.: 1612188-96-1
Target:  

Neurotensin Receptor

Research Areas:  

Neurological Disease

NTRC-739 is a selective nonpeptide partial neurotensin receptor type 2 (NTS2) agonist with an EC50 of 12 nM and a Ki of 153 nM. NTRC-739 is 161-fold selective for NTS2 versus NTS1. NTRC-739 can be used for the study of chronic pain research .
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