Sepimostat dimethanesulfonate
Based on 2 publication(s) in Google Scholar
Sepimostat dimethanesulfonate (FUT-187) exhibits neuroprotective activity via NR2B N-methyl-D-aspartate receptor antagonism at the Ifenprodil-binding site of the NR2B subunit. Sepimostat dimethanesulfonate inhibits the Ifenprodil binding with a Ki value of 27.7 µM.
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- CAS No.: 103926-82-5
- Formule: C23H27N5O8S2
- Masse moléculaire:565.62
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Activité biologique
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
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Animal Model:Male Sprague Dawley rats weighing 150-300 g[1].
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Dosage:Intravitreal injection.
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Administration:1 to 100 nmol/eye.
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Result:Exhibited neuroprotective effects significantly.
Chemical Information
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CAS No. 103926-82-5
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Masse moléculaire 565.62
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Formule C23H27N5O8S2
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SMILES
O=C(OC1=CC=C2C=C(C(N)=N)C=CC2=C1)C3=CC=C(NC4=NCCN4)C=C3.CS(=O)(O)=O.CS(=O)(O)=O
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Synonyms
FUT-187
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Publications (2)
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Journal Impact Factor
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Most Recent
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Eur J Pharmacol
Mechanisms of acid-sensing ion channels inhibition by nafamostat, sepimostat and diminazene. [Abstract]2023 Jan 5:938:175394. PMID: 36403685 -
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Sepimostat dimethanesulfonate Related Classifications
HY-136299A Related Classifications
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