TM38837
TM38837 is an orally active and selective inverse agonist of cannabinoid receptor 1 (CB1) with an IC50 of 24 nM. TM38837 has higher selectivity for CB1 than for CB2 (IC50: 4500 nM). TM38837 can reduce body weight, improve plasma inflammatory markers and glucose homeostasis.
For research use only. We do not sell to patients.
- CAS No.: 1034264-77-1
- Formula: C27H20Cl2F3N7O
- Molecular Weight:586.40
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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CB1 |
Chemical Information
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CAS No. 1034264-77-1
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Molecular Weight 586.40
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Formula C27H20Cl2F3N7O
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SMILES
FC(F)(C1=CC=C([C@@H](C)NC(C2=NN(C3=CC=CC=C3Cl)C(C4=CC=C(Cl)C=C4)=C2CC5=NNN=N5)=O)C=C1)F
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)