2. Membrane Transporter/Ion Channel Neuronal Signaling
  3. TRP Channel
  4. TRPV1 antagonist 6

TRPV1 antagonist 6 (compound 51) is a mode-selective antagonist for transient receptor potential vanilloid member 1 (TRPV1), which shows antagonism with IC50 of 2.85 nM to capsaicin activation and 28.48 % inhibition against proton activation at a 3 µM concentration.

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TRPV1 antagonist 6

TRPV1 antagonist 6 Estructura química

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TRPV1 antagonist 6 Related Antibodies

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Descripciòn

TRPV1 antagonist 6 (compound 51) is a mode-selective antagonist for transient receptor potential vanilloid member 1 (TRPV1), which shows antagonism with IC50 of 2.85 nM to capsaicin activation and 28.48 % inhibition against proton activation at a 3 µM concentration[1].

Peso molecular

493.99

Fòrmula

C26H28ClN5O3
SMILES

CC(C)(C)C1=NN(C(CNC(NC2=CC=CC(N3CCO)=C2C=CC3=O)=O)=C1)C4=CC=CC(Cl)=C4
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TRPV1 antagonist 6 Related Classifications

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Keywords:

TRPV1 antagonist 6TRP ChannelTransient receptor potential channelsVanilloid Receptor 1capsaicin and heat activated nociceptorInhibitorinhibitorinhibit

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TRPV1 antagonist 6
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HY-161273
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