1. Antibody-drug Conjugate/ADC Related
  2. ADC Linker
  3. Vipivotide tetraxetan Linker

Vipivotide tetraxetan Linker (Synonyms: PSMA-617 Linker)

Cat. No.: HY-43869
Handling Instructions

Vipivotide tetraxetan Linker is a useful peptide linker for synthesis of Vipivotide tetraxetan (PSMA-617). Vipivotide tetraxetan (PSMA-617) is a ligand used to synthesize 177Lu-PSMA-617, which is a radioactive molecule for the treatment of prostate cancer.

For research use only. We do not sell to patients.

Vipivotide tetraxetan Linker Chemical Structure

Vipivotide tetraxetan Linker Chemical Structure

CAS No. : 1703768-74-4

Size Price Stock Quantity
10 mM * 1 mL in DMSO USD 2200 In-stock
Estimated Time of Arrival: December 31
50 mg USD 2000 In-stock
Estimated Time of Arrival: December 31
100 mg USD 3500 In-stock
Estimated Time of Arrival: December 31
250 mg USD 6500 In-stock
Estimated Time of Arrival: December 31
500 mg   Get quote  
1 g   Get quote  

* Please select Quantity before adding items.

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Based on 1 publication(s) in Google Scholar

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Description

Vipivotide tetraxetan Linker is a useful peptide linker for synthesis of Vipivotide tetraxetan (PSMA-617). Vipivotide tetraxetan (PSMA-617) is a ligand used to synthesize 177Lu-PSMA-617, which is a radioactive molecule for the treatment of prostate cancer[1].

IC50 & Target

Alkyl-Chain

 

Molecular Weight

655.74

Formula

C₃₃H₄₅N₅O₉

CAS No.

1703768-74-4

SMILES

O=C(O)[[email protected]](CCCCNC([[email protected]](CC1=CC=C2C=CC=CC2=C1)NC([[email protected]]3CC[[email protected]](CN)CC3)=O)=O)NC(N[[email protected]](C(O)=O)CCC(O)=O)=O

Shipping

Room temperature in continental US; may vary elsewhere

Storage
Powder -80°C 2 years
  -20°C 1 year
In solvent -80°C 6 months
  -20°C 1 month
Solvent & Solubility
In Vitro: 

DMSO : 270 mg/mL (411.75 mM; Need ultrasonic)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 1.5250 mL 7.6250 mL 15.2499 mL
5 mM 0.3050 mL 1.5250 mL 3.0500 mL
10 mM 0.1525 mL 0.7625 mL 1.5250 mL
*Please refer to the solubility information to select the appropriate solvent.
In Vivo:
  • 1.

    Add each solvent one by one:  10% DMSO    40% PEG300    5% Tween-80    45% saline

    Solubility: ≥ 2.25 mg/mL (3.43 mM); Clear solution

  • 2.

    Add each solvent one by one:  10% DMSO    90% (20% SBE-β-CD in saline)

    Solubility: ≥ 2.25 mg/mL (3.43 mM); Clear solution

  • 3.

    Add each solvent one by one:  10% DMSO    90% corn oil

    Solubility: ≥ 2.25 mg/mL (3.43 mM); Clear solution

*All of the co-solvents are provided by MCE.
References
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Product Name:
Vipivotide tetraxetan Linker
Cat. No.:
HY-43869
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