1. Metabolic Enzyme/Protease
  2. Dipeptidyl Peptidase
  3. Dutogliptin

Dutogliptin (Synonyms: PHX-1149 free base)

Cat. No.: HY-10286
Handling Instructions

Dutogliptin (PHX-1149 free base) is an orally available, potent, and selective dipeptidyl peptidase-4 (DPP4) inhibitor for the treatment of type 2 diabetes mellitus.

For research use only. We do not sell to patients.

Dutogliptin Chemical Structure

Dutogliptin Chemical Structure

CAS No. : 852329-66-9

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Description

Dutogliptin (PHX-1149 free base) is an orally available, potent, and selective dipeptidyl peptidase-4 (DPP4) inhibitor for the treatment of type 2 diabetes mellitus.

IC50 & Target

DPP4[1]

In Vivo

Dutogliptin exhibits low plasma protein binding (11%) and is rapidly absorbed with a Tmax of 3-4 h and a half-life of 10-13 h. Dutogliptin is metabolically stable and does not inhibit or induce the activity of major CYP450s[2].

Clinical Trial
Molecular Weight

241.10

Formula

C₁₀H₂₀BN₃O₃

CAS No.

852329-66-9

SMILES

O=C(CN[[email protected]@H]1CCNC1)N(CCC2)[[email protected]@H]2B(O)O

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Keywords:

DutogliptinPHX-1149PHX1149PHX 1149Dipeptidyl PeptidaseDPPDPP4diabetesmellitusInhibitorinhibitorinhibit

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