1. Metabolic Enzyme/Protease
    Anti-infection
  2. HIV Integrase
    HIV

HIV-1 integrase inhibitor 4 

Cat. No.: HY-108820
Handling Instructions

HIV-1 integrase inhibitor 4 is a HIV-1 integrase strand transfer (INST) inhibitor with an IC50 of 3.7 nM.

For research use only. We do not sell to patients.

HIV-1 integrase inhibitor 4 Chemical Structure

HIV-1 integrase inhibitor 4 Chemical Structure

CAS No. : 1638504-66-1

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  • Biological Activity

  • Technical Information

  • Purity & Documentation

  • References

Description

HIV-1 integrase inhibitor 4 is a HIV-1 integrase strand transfer (INST) inhibitor with an IC50 of 3.7 nM.

IC50 & Target

IC50: 3.7 nM (INST)[1]

In Vitro

HIV-1 integrase inhibitor 4 (compound 4f) is a HIV-1 integrase strand transfer (INST) inhibitor with an IC50 of 3.7 nM. HIV-1 integrase inhibitor 4 shows potent activity against recombinant HIV IN in biochemical assays and good efficacy in assays done in cell culture against a broad panel of viral mutants carrying the major RAL and DTG IN resistance mutations[1].

References
Molecular Weight

514.50

Formula

C₂₄H₂₀F₂N₄O₅S

CAS No.

1638504-66-1

SMILES

NC(C1=CC(CCS(=O)(C2=CC=CC=C2)=O)=CN=C1N3O)=C(C(NCC4=CC=C(F)C=C4F)=O)C3=O

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Shipping

Room temperature in continental US; may vary elsewhere

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

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Product Name:
HIV-1 integrase inhibitor 4
Cat. No.:
HY-108820
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HIV-1 integrase inhibitor 4

Cat. No.: HY-108820