2. Others

Others (その他)

Others

関連製品

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There are a number of inhibitors, agonists, and antagonists which we cannot make precise classification because the research area is still unknown.

Others 関連製品 (73921):

製品番号 製品名 CAS 番号 純度 構造式
  • HY-136504
    Bianthrone 434-85-5 98%
    Bianthrone (Dianthrone) is a natural product that can be isolated from Rheum officinale Baill. Bianthrone is a potential toxic marker of Polygonum multiflorum Thunb.
    Bianthrone
  • HY-136513S
    Bifenox-d3 98%
    Bifenox-d3 is the deuterium labeled Bifenox. Bifenox (MC-4379) is a nitrophenyl ether herbicide. Bifenox disrupts cellular membrane, inhibits photosynthesis and inhibits the protoporphyrinogen oxidase. Bifenox increases the ROS production in the microalgae Chlamydomonas reinhardtii.
    Bifenox-d3
  • HY-136612R
    DCBA (Standard) 72236-23-8
    Pteroic acid (Standard) is the analytical standard of Pteroic acid. This product is intended for research and analytical applications. Pteroic acid is an active compound.
    DCBA (Standard)
  • HY-136614
    H-Val-βNA 729-24-8 98%
    H-Val-βNA (L-Valine β-naphthylamide) can be used as an aminopeptidase and a Valine arylamidase substrate.
    H-Val-βNA
  • HY-136628
    RU 25434 62622-76-8 98%
    RU 25434 is an active compound.
    RU 25434
  • HY-136630
    Felotaxel 944154-59-0 98%
    Felotaxel (SHR110008) is a derivate of Docetaxel (HY-B0011), with antitumor activity and specific pharmacokinetic properties in rats. Felotaxel is rapidly distributed to normal tissues. The kidney is the major excretion organ, and its plasma protein binding capacity is nearly linearly related to concentration.
    Felotaxel
  • HY-136634
    BTM-1042 72293-40-4 98%
    BTM-1042 is a newly synthesized compound with antispasmodic effects. It can inhibit the twitch reaction of the guinea pig ileum under electrical stimulation and is not affected by naloxone. It has similar effects to atropine and can block muscarinic receptors, but has less effect on other types of receptors. BTM-1042 also has an inhibitory effect on the ileal reaction caused by nicotine and 5-hydroxytryptamine. BTM-1042 showed a dose-dependent inhibitory effect on the spontaneous movement of the rabbit stomach. In general, BTM-1042 is a agent with a strong antispasmodic effect.
    BTM-1042
  • HY-136644
    PD-217014-methyl ester 444088-20-4 98%
    PD-217014-methyl ester is an α?δ ligand with visceral analgesic activity and can inhibit visceral hypersensitivity, and its anti-hyperalgesic effect is dose-dependent.
    PD-217014-methyl ester
  • HY-136644A
    PD-217014 335458-65-6 98%
    PD-217014 is an α2δ ligand with visceral analgesic activity and can inhibit visceral hypersensitivity reactions. Its anti-allodynic effect is dose-dependent.
    PD-217014
  • HY-136648S
    2'-Deoxyadenosine-5'-triphosphate-13C10,15N5 (tetraammonia) 98%
    2'-Deoxyadenosine-5'-triphosphate-13C10,15N5 tetraammonia is the 13C10 and 15N5 labeled 2'-Deoxyadenosine-5'-triphosphate (HY-136648). 2'-Deoxyadenosine-5'-triphosphate (dATP) is a nucleotide used in cells for DNA synthesis (or replication), as a substrate of DNA polymerase.
    2'-Deoxyadenosine-5'-triphosphate-13C10,15N5 (tetraammonia)
  • HY-136648S2
    2'-Deoxyadenosine-5'-triphosphate-15N5,d14 dilithium 98%
    2'-Deoxyadenosine-5'-triphosphate-15N5,d14 (dATP-15N5,d14) dilithium is deuterium and 15N labeled 2'-Deoxyadenosine-5'-triphosphate (HY-136648). 2'-Deoxyadenosine-5'-triphosphate (dATP) is a nucleotide used in cells for DNA synthesis (or replication), as a substrate of DNA polymerase.
    2'-Deoxyadenosine-5'-triphosphate-15N5,d14 dilithium
  • HY-136648S4
    2'-Deoxyadenosine-5'-triphosphate-15N5 dilithium 99.30%
    2'-Deoxyadenosine-5'-triphosphate-15N5 (dATP-15N5) dilithium is 15N labeled 2'-Deoxyadenosine-5'-triphosphate (HY-136648). 2'-Deoxyadenosine-5'-triphosphate (dATP) is a nucleotide used in cells for DNA synthesis (or replication), as a substrate of DNA polymerase.
    2'-Deoxyadenosine-5'-triphosphate-15N5 dilithium
  • HY-136648S5
    2'-Deoxyadenosine-5'-triphosphate-13C10 dilithium
    2'-Deoxyadenosine-5'-triphosphate-13C10 (dATP-13C10) dilithium is 13C-labeled 2'-Deoxyadenosine-5'-triphosphate (HY-136648). 2'-Deoxyadenosine-5'-triphosphate (dATP) is a nucleotide used in cells for DNA synthesis (or replication), as a substrate of DNA polymerase.
    2'-Deoxyadenosine-5'-triphosphate-13C10 dilithium
  • HY-136649
    2'-Deoxy-2'-fluoroadenosine 5'-triphosphate tetralithium 98%
    2'-Deoxy-2'-fluoroadenosine 5'-triphosphate tetralithium is an ATP analog, it exerted a strong but mixed-type inhibition on poly(AU) synthesis.
    2'-Deoxy-2'-fluoroadenosine 5'-triphosphate tetralithium
  • HY-136659
    Ro 04-5595 194089-07-1 98%
    Ro 04-5595 is a selective antagonist with specific activity against the NR2B subunit of the NMDA receptor. Ro 04-5595 exhibits favorable pharmacokinetic properties in in vitro and in vivo studies, with rapid uptake and clearance. Ro 04-5595 exhibits strong binding in NR2B receptor-enriched regions and low binding in the cerebellum. Ro 04-5595 is able to effectively inhibit specific binding, showing high affinity for the NR2B receptor and a clear ranking of binding affinity with a variety of other compounds.
    Ro 04-5595
  • HY-136675
    ASMI 1850419-05-4 98%
    ASMI is a ratiometric, two-photon excited fluorescent probe, composed of a highly two-photon active and biocompatible merocyanine fluorophore and an acrylate moiety as a thiol reactive site. ASMI is able to selectively detect and monitor mitochondrial Cys with rapid responsiveness, imaging living cells and intact tissues with high contrast and brightness at a depth of 150 μm. The two-photon action cross section (Φσmax) of ASMI is 65.2 GM, corresponding to an excitation wavelength (λex) of 740 nm.
    ASMI
  • HY-136690
    Triasulfuron 82097-50-5 98%
    Triasulfuron is a sulfonylurea herbicide. Triasulfuron degrades slowly, with most of the residues remaining in the first 20 cm of the soil surface, but small amounts have been observed to penetrate deeper into the soil (up to 1 m deep).
    Triasulfuron
  • HY-136720
    ZXX2-77 304913-22-2 98%
    ZXX2-77 is a cyclooxygenase-1 (COX-1) selective inhibitor belonging to the benzenesulfonylanilide class of compounds. It is reported as a novel analgesic that does not cause gastric damage. ZXX2-77 has a weak analgesic effect but exhibits potent COX-1 inhibitory activity in vitro. The low oral absorption rate of ZXX2-77 leads to its weak analgesic effect in vivo. At a dose of 30 mg/kg, the maximum plasma concentration of ZXX2-77 (1.2 mM) did not reach its COX-1 IC50 value (3.2 mM). In contrast, its derivative ZXX2-79, although weaker in vitro COX inhibitory activity, is better absorbed, exhibits stronger analgesic effect and hardly causes gastric damage. These findings suggest that ZXX2-77 and its derivatives as COX-1 selective inhibitors may become effective analgesics that do not cause gastric damage.
    ZXX2-77
  • HY-136779S
    Antioxidant 245-d12
    Antioxidant 245-d12 (AO-245-d12) is the deuterium labeled Antioxidant 245 (HY-136779). Antioxidant 245 (AO-245) is a hindered phenol antioxidant. Antioxidant 245 can be used in the research of nanocomposites.
    Antioxidant 245-d12
  • HY-136784
    Rhod-2 potassium 663625-18-1 98%
    Rhod-2 potassium is a cell impermeant, red fluorescent calcium indicator. Rhod-2 potassium exhibits a significant shift in fluorescence intensity upon calcium binding (ex max=549 nm; calcium-free v. ex/em max=552/581 nm; calcium-bound). Unlike the UV-excitable indicators Fura-2 and Indo-1 (HY-D0121), there is no accompanying spectral shift.
    Rhod-2 potassium