1. GPCR/G Protein
  2. Sigma Receptor
  3. Sigma-2 receptor antagonist 1

Sigma-2 receptor antagonist 1 

Cat. No.: HY-111669
Handling Instructions

Sigma-2 receptor antagonist 1 is a sigma-2 (σ-2) receptor antagonist.

For research use only. We do not sell to patients.

Sigma-2 receptor antagonist 1 Chemical Structure

Sigma-2 receptor antagonist 1 Chemical Structure

CAS No. : 1802632-22-9

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Description

Sigma-2 receptor antagonist 1 is a sigma-2 (σ-2) receptor antagonist.

IC50 & Target

Sigma-2 receptor

Molecular Weight

431.59

Formula

C₂₄H₃₃NO₄S

CAS No.

1802632-22-9

SMILES

OC1=CC=C(CCC(C)(N2CC3=C(C=C(S(=O)(C)=O)C=C3)C2)C)C=C1OC(C)(C)C

Shipping

Room temperature in continental US; may vary elsewhere

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Solvent & Solubility
In Vitro: 

DMSO : 250 mg/mL (579.25 mM; Need ultrasonic)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.3170 mL 11.5851 mL 23.1701 mL
5 mM 0.4634 mL 2.3170 mL 4.6340 mL
10 mM 0.2317 mL 1.1585 mL 2.3170 mL
*Please refer to the solubility information to select the appropriate solvent.
In Vivo:
  • 1.

    Add each solvent one by one:  10% DMSO    40% PEG300    5% Tween-80    45% saline

    Solubility: ≥ 2.08 mg/mL (4.82 mM); Clear solution

  • 2.

    Add each solvent one by one:  10% DMSO    90% (20% SBE-β-CD in saline)

    Solubility: ≥ 2.08 mg/mL (4.82 mM); Clear solution

  • 3.

    Add each solvent one by one:  10% DMSO    90% corn oil

    Solubility: ≥ 2.08 mg/mL (4.82 mM); Clear solution

*All of the co-solvents are provided by MCE.
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Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

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Product Name:
Sigma-2 receptor antagonist 1
Cat. No.:
HY-111669
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