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Cannabinoid Receptor Related Products (294)
Related Products (294)
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(1H-Indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone
0 ImagesSynonyms: UR-144 Impurity 3(1H-Indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone (UR-144 Impurity 3) is a precursor in the synthesis of synthetic cannabinoids.
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Linoleoyl ethanolamide-d4
0 ImagesLinoleoyl ethanolamide-d4 is a deuterated labeled Linoleoyl ethanolamide. Linoleoyl ethanolamide (Linoleic acid monoethanolamide) is classified as a fatty acid ethanolamide. Linoleoyl ethanolamide only weakly binds G-protein-coupled cannabinoid receptors of type-1（CB1）and CB2 receptors, and inhibits the binding of [3H]CP-55,940 with Kis of 10 and 25 μM, respectively. Linoleoyl ethanolamide is 4-fold less potent than anandamide at causing catalepsy in mice and it does not prolong sleep time.
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A-836339
0 ImagesA-836339 is a selective CB2 receptor agonist, with Ki values of 0.4 nM and 0.8 nM in humans and rats, respectively. A-836339 exhibits multiple effects such as analgesia, gastric protection, anti-inflammation, and antioxidant activity. A-836339 produces antinociceptive and analgesic activities by activating CB2 receptors in the dorsal root ganglia and spinal cord. A-836339 can also exert gastric protective effects through anti-inflammatory mechanisms (reducing TNF-α and IL-1β) and antioxidant mechanisms (enhancing the activities of CAT and SOD, and reducing H2O2). Radioactively labeled A-836339 can serve as a CB2-specific radioligand for autoradiography and PET imaging. A-836339 can be used in research on inflammatory pain, neuropathic pain, gastric ulcers, cerebral ischemia, etc.
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Pregnenolone monosulfate-d4 sodium
0 ImagesSynonyms: 3β-Hydroxy-5-pregnen-20-one monosulfate-d4 sodiumPregnenolone monosulfate-d4 sodium is the deuterium labeled Pregnenolone monosulfate sodium (HY-110189) . Pregnenolone monosulfate sodium (3β-Hydroxy-5-pregnen-20-one monosulfate sodium) is a powerful neurosteroid, the main precursor of various steroid hormones including steroid ketones. Pregnenolone monosulfate sodium acts as a signaling-specific inhibitor of cannabinoid CB1 receptor, inhibits the effects of tetrahydrocannabinol (THC) that are mediated by the CB1 receptors. Pregnenolone monosulfate sodium can protect the brain from cannabis intoxication. Pregnenolone monosulfate sodium is also a TRPM3 channel activator, and also can weakly activate TRPM1 channels.
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6α-Hydroxy-cannabidiol
0 ImagesSynonyms: 6α-OH-CBD6α-Hydroxy-cannabidiol (6α-OH-CBD) is a metabolite of Cannabidiol.
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Pregnenolone-d4
0 ImagesCat. No.: HY-B0151SSynonyms: 3β-Hydroxy-5-pregnen-20-one-d4Pregnenolone-d4 is the deuterium labeled Pregnenolone. Pregnenolone (3β-Hydroxy-5-pregnen-20-one) is a powerful neurosteroid, the main precursor of various steroid hormones including steroid ketones. Pregnenolone acts as a signaling-specific inhibitor of cannabinoid CB1 receptor, inhibits the effects of tetrahydrocannabinol (THC) that are mediated by the CB1 receptors. Pregnenolone can protect the brain from cannabis intoxication. Pregnenolone is also a TRPM3 channel activator, and also can weakly activate TRPM1 channels.
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Hemopressin(rat)
0 ImagesHemopressin(rat) is a nonapeptide derived from the α1-chain of hemoglobin, is originally isolated from rat brain homogenates. Hemopressin(rat) is orally active, selective and inverse agonist of CB1 cannabinoid receptors. Hemopressin(rat) exerts antinociceptive action in inflammatory pain models.
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Arachidonoyl ethanolamide phosphate
0 ImagesCat. No.: HY-134173CAS No.: 183323-26-4
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(R)-JD-5037
0 ImagesCat. No.: HY-18697ACAS No.: 1404117-65-2
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10(R)-Hydroxy-9(S)-hexahydrocannabinol
0 ImagesCat. No.: HY-170043ACAS No.: 60948-21-210(R)-Hydroxy-9(S)-hexahydrocannabinol is structurally similar to known phytocannabinoids.
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b-AEA
0 ImagesCat. No.: HY-103329CAS No.: 956605-71-3Synonyms: MM22; Biotinylated N-arachidonoylethanolamineb-AEA (MM22) is a biotinylated endocannabinoid analog with probe activity. b-AEA is able to accumulate intracellularly in a similar manner to the parent compound AEA. b-AEA does not interact with other components of the endocannabinoid system and therefore does not interfere with their function. b-AEA can be used to visualize the accumulation and intracellular distribution of endocannabinoids.
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Cannabidiol-C8
0 ImagesCat. No.: HY-170734CAS No.: 2552798-28-2Cannabidiol-C8 is structurally similar to known phytocannabinoids.
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Cannabinodiol
0 ImagesCannabinodiol, a cannabinoid analogue, is a phytocannabinoid.
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OMDM-6
0 ImagesCat. No.: HY-135882CAS No.: 616884-67-4OMDM-6 is a hybrid agonist of vanilloid receptor type 1 (VR1, TRPV1) (EC50=75 nM) and cannabinoid receptor type 1 (CB1) (Ki=3.2 μM). OMDM-6 inhibits anandamide cellular uptake (ACU) with a Ki of 7.0 μM.
