2. Signaling Pathways
  3. GPCR/G Protein
  4. G protein-coupled Bile Acid Receptor 1
  5. G protein-coupled Bile Acid Receptor 1 Antagonist

G protein-coupled Bile Acid Receptor 1 Antagonist

G protein-coupled Bile Acid Receptor 1 Antagonists (3):

Cat. No. Product Name Effect Purity
  • HY-111534
    SBI-115
    		Antagonist 99.69%
    SBI-115 is a TGR5 (GPCR19) antagonist. SBI-115 decreases hepatic cystogenesis with polycystic liver diseases via inhibiting TGR5.
  • HY-139677A
    5-HT7R antagonist 1 free base
    		Antagonist
    5-HT7R antagonist 1 (free base) is a G protein-biased antagonist against 5-HT7R (Ki = 6.5 nM).
  • HY-139677
    5-HT7R antagonist 1
    		Antagonist
    5-HT7R antagonist 1 is a G protein-biased antagonist against 5-HT7R (Ki = 6.5 nM).