AHR antagonist 4
AHR antagonist 4 is a 2-heteroaryl-3-oxo-2,3-dihydropyridazine-4-carboxamide compound and a potent aryl hydrocarbon receptor (AHR) antagonist extracted from patent WO2018146010A1, example 293, has an IC50 of 82.2 nM. AHR antagonist 4 has anti-cancer effects.
For research use only. We do not sell to patients.
- CAS No.: 2242465-58-1
- Formula: C20H14F6N4O4
- Molecular Weight:488.34
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
IC50: 82.2 nM (Aryl hydrocarbon receptor (AHR))[1]
Chemical Information
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CAS No. 2242465-58-1
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Molecular Weight 488.34
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Formula C20H14F6N4O4
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SMILES
O=C(C1=CC(C2=CC=C(OC(F)(F)F)C=C2)=NN(C3=CC=CN=C3)C1=O)NC[C@H](O)C(F)(F)F
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)