AR antagonist 7
AR antagonist 7 (86) is an androgen receptor (AR) antagonist that can be used in the research of hair loss.
For research use only. We do not sell to patients.
- CAS No.: 876759-97-6
- Formula: C16H12F3NO2
- Molecular Weight:307.27
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Size
Price
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
Description
AR antagonist 7 (86) is an androgen receptor (AR) antagonist that can be used in the research of hair loss[1].
Cellular Effect
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| MDA-MB-231 | IC50 |
299 nM
Compound: 6l
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Antagonist activity at human androgen receptor expressed in human MDA-MB-231 cells assessed as inhibition of DHT-induced response
Antagonist activity at human androgen receptor expressed in human MDA-MB-231 cells assessed as inhibition of DHT-induced response
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[PMID: 19286380] |
| Sf9 | IC50 |
69 nM
Compound: 6l
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Displacement of [3H]DHT from human cloned androgen receptor expressed in insect Sf9 cell system
Displacement of [3H]DHT from human cloned androgen receptor expressed in insect Sf9 cell system
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[PMID: 19286380] |
Chemical Information
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CAS No. 876759-97-6
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Molecular Weight 307.27
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Formula C16H12F3NO2
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SMILES
N#CC1=CC=C(OC2=CC=C(C)C=C2OC)C=C1C(F)(F)F
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
Select Batch:
Purity:
99.98%
Assay:
99.98%
ee.:
99.98%
References
Calculators
Molarity Calculator
Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)
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Dilution Calculator
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