AR ligand-49
AR ligand-49 (Compound 4q) is a dual ligand for the adenosine A2A receptor (A2AAR) and the A3 receptor (A3AR). Its Ki values are 15 and 4.5 nM respectively. AR ligand-49 exhibits reverse agonistic activity at hA2AAR and antagonistic activity at hA3AR. AR ligand-49 can be used for the study of the design and development of adenosine receptor ligands.
For research use only. We do not sell to patients.
- Formula: C19H23N7O3S
- Molecular Weight:429.50
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
Chemical Information
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Molecular Weight 429.50
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Formula C19H23N7O3S
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SMILES
NC1=NC(NC2=C(N3CCOCC3)C=CC=C2)=NC4=C1N=CN4[C@@H]5SC[C@@H](O)[C@H]5O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)