BMS-986034
BMS-986034 is an orally active ingredient (API) that is an agonist of GPR119..
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- CAS. Nr.: 1492631-88-5
- Formel: C24H24Cl2N6O4
- Molecular Weight:531.39
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Speicherung:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biologische Aktivität
GPR119[1]
|
Cell Line
|
Type | Value | Description | References |
|---|---|---|---|---|
| HEK293 | EC50 |
3 nM
Compound: 4
|
Agonist activity at human-mouse chimeric GPR119 expressed in tetracycline-induced Flp-In-T-Rex-HEK293 cells assessed as accumulation of cAMP after 50 mins by HTRF assay
Agonist activity at human-mouse chimeric GPR119 expressed in tetracycline-induced Flp-In-T-Rex-HEK293 cells assessed as accumulation of cAMP after 50 mins by HTRF assay
|
[PMID: 24900860] |
Chemical Information
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CAS. Nr. 1492631-88-5
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Molecular Weight 531.39
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Formel C24H24Cl2N6O4
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SMILES
O=C1C=C(C(Cl)=CN1C2=NC(C)=C(C=C2)N3C([C@@H](CC3)O)=O)OC4CCN(CC4)C5=NC=C(C=N5)Cl
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Versand
Room temperature in continental US; may vary elsewhere.
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Speicherung
Please store the product under the recommended conditions in the Certificate of Analysis.
Reinheit & Dokumentation
Verweise
Calculators
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)