IUN-00433
IUN-00433 (Compound 36) is a selective positive allosteric modulator of α4β1δ-type GABAA receptors, with an EC50 of 0.060 μM. IUN-00433 is applicable to research related to neurological disorders.
For research use only. We do not sell to patients.
- CAS No.: 2188230-70-6
- Formula: C18H11BrClN3OS
- Molecular Weight:432.72
-
Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
-
Biological Activity
-
Chemical Information
- Purity & Documentation
- References
-
Help & FAQs
Biological Activity
|
α4β1δ GABAA 0.060 μM (EC50) |
IUN-00433 exerts positive allosteric regulatory activity on α4β1δ, with an EC50 of 0.060 μM, which is 16-fold more potent than DS2[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
-
CAS No. 2188230-70-6
-
Molecular Weight 432.72
-
Formula C18H11BrClN3OS
-
SMILES
O=C(C1=CC=C(C=C1)Cl)NC2=C(C3=CC=CS3)N=C4C=CC(Br)=CN42
-
Shipping
Room temperature in continental US; may vary elsewhere.
-
Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
IUN-00433 Related Classifications
HY-182511 Related Classifications
Powered by Bioz