PREP-IN-2
PREP-IN-2 is an irreversible and selective prolyl endopeptidase (PREP) inhibitor with an IC50 of 0.53 μM and a Ki of 0.62 μM. PREP-IN-2 can be used in research related to neurodegenerative diseases and triple-negative breast cancer.
For research use only. We do not sell to patients.
- Formula: C22H24ClN5O2
- Molecular Weight:425.91
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
PREP-IN-2 (Compound 14) (0.001-10 μM; 4 h) inhibits PREP activity in SH-SY5Y and MDA-MB-231 cells, with IC50 values of 67 nM and 127 nM, respectively[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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Molecular Weight 425.91
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Formula C22H24ClN5O2
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SMILES
ClC1=C(C(NCC(N2CCCC2)=O)=O)C=NC3=C1C(C)=NN3CCC4=CC=CC=C4
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
PREP-IN-2 Related Classifications
HY-181070 Related Classifications
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