IUN-00433
IUN-00433 (Compound 36) is a selective positive allosteric modulator of α4β1δ-type GABAA receptors, with an EC50 of 0.060 μM. IUN-00433 is applicable to research related to neurological disorders.
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- CAS No.: 2188230-70-6
- Formule: C18H11BrClN3OS
- Masse moléculaire:432.72
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Activité biologique
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α4β1δ GABAA 0.060 μM (EC50) |
IUN-00433 exerts positive allosteric regulatory activity on α4β1δ, with an EC50 of 0.060 μM, which is 16-fold more potent than DS2[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 2188230-70-6
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Masse moléculaire 432.72
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Formule C18H11BrClN3OS
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SMILES
O=C(C1=CC=C(C=C1)Cl)NC2=C(C3=CC=CS3)N=C4C=CC(Br)=CN42
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)