TD-5471
TD-5471 is a potent and selective full agonist of the human β2-adrenoceptor.
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- CAS No.: 530084-87-8
- Formule: C32H31N3O4
- Masse moléculaire:521.61
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Activité biologique
β2 adrenoceptor[1]
TD-5471 is potent, with slow onset in an in vitro guinea pig trachea model. TD-5471 has potency with pEC50 of 8.7 in the guinea pig tracheal ring assay.TD-5471 is structurally differentiated from Milveterol (HY-14297) and its long duration of action is consistent with a correlation with hydrophobicity observed in other long-acting β2-agonist discovery programs[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 530084-87-8
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Masse moléculaire 521.61
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Formule C32H31N3O4
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SMILES
O=C1NC2=C(C([C@@H](O)CNCCC3=CC=C(NC4=CC(C5=CC=CC=C5)=C(OC)C=C4)C=C3)=CC=C2O)C=C1
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)