1083076-69-0
1083076-69-0
Chemical Structure
Cariprazine hydrochloride
Synonym(s): RGH188 hydrochloride
- CAS No.: 1083076-69-0
- Formula:C21H33Cl3N4O
- Molecular Weight:463.87
IUPAC Name: 3-((1r,4r)-4-(2-(4-(2,3-dichlorophenyl)piperazin-1-yl)ethyl)cyclohexyl)-1,1-dimethylurea hydrochloride
InChIKey: GPPJWWMREQHLQT-BHQIMSFRSA-N
SMILES: O=C(N[C@H]1CC[C@H](CCN2CCN(C3=CC=CC(Cl)=C3Cl)CC2)CC1)N(C)C.[H]Cl
Biological Activity: Cariprazine hydrochloride is a novel antipsychotic agent candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (Ki=2.6 nM).
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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Cariprazine hydrochloride | 99.88% | Cariprazine hydrochloride is a novel antipsychotic agent candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (Ki=2.6 nM). | ||||||||||||||||||||
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Structural Analogs
-
Similarity Score 0.98
HY-14763RCariprazine (Standard) -
Similarity Score 0.88
HY-100656RDesmethyl cariprazine (Standard) -
Similarity Score 0.88
HY-100658RDidesmethyl cariprazine (Standard) -
Similarity Score 0.86
HY-177122Raxlaprazine etomoxil -
Similarity Score 0.83
HY-183776Dopamine D3 receptor agonist-2 -
Similarity Score 0.82
HY-156239Dopamine D3 receptor ligand-5 -
Similarity Score 0.82
HY-W724128Cariprazine N-oxide -
Similarity Score 0.81
HY-14763SCariprazine-d6 -
Similarity Score 0.79
HY-47412Cariprazine impurity 1 -
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