Cariprazine impurity 1
Based on 1 Customer Validation
Cariprazine impurity 1 is a dopamine D2 receptor (D2R) agonist. Cariprazine impurity 1 modulates D2R-mediated Gi/o signaling pathway to inhibit cAMP production, and regulates D2R-mediated β-arrestin2 recruitment pathway.
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研究用途以外に使用した場合、当社は一切の責任を負いかねます。
- CAS 番号: 791778-53-5
- 分子式: C18H27Cl2N3
- 分子量:356.34
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保管条件:
4°C, protect from light
* In solvent : -80°C, 6 months; -20°C, 1 month (protect from light)
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生物活性
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化学情報
- 純度とドキュメンテーション
- 参考文献
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Help & FAQs
Dopamine Receptor アイソフォーム固有の製品をすべて表示
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生物活性
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D2 Receptor |
Cariprazine impurity 1 (Compound 11) acts as a balanced partial agonist of human D2R, mediates Gi/o-dependent cAMP inhibition (with an EC50 of 0.7 nM) and β-arrestin2 recruitment (with an EC50 of 2 nM), and exhibits a mild bias toward the Gi/o signaling pathway[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
化学情報
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CAS 番号 791778-53-5
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性状 Solid
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分子量 356.34
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分子式 C18H27Cl2N3
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SMILES
ClC1=C(N2CCN(CC[C@H]3CC[C@H](N)CC3)CC2)C=CC=C1Cl
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
4°C, protect from light
* In solvent : -80°C, 6 months; -20°C, 1 month (protect from light)
純度とドキュメンテーション
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データシート (266 KB)
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SDS (393 KB)
- English - EN (393 KB)
- Français - FR (393 KB)
- Deutsch - DE (393 KB)
- Norwegian - NO (393 KB)
- Español - ES (393 KB)
- Swedish - SV (393 KB)
- Italian - IT (393 KB)
- Korean - KR (393 KB)
- Portuguese - PT (393 KB)
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取扱説明書 (2659 KB)
参考文献
Calculators
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)
Cariprazine impurity 1 関連分類
HY-47412 関連分類
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