2. GPCR/G Protein
    Neuronal Signaling
  3. Dopamine Receptor
    5-HT Receptor
  4. Cariprazine-d6

Cariprazine-d6  (Synonyms: RGH-188-d6)

Cat. No.: HY-14763S Purity: 98.00%
COA Handling Instructions

Cariprazine-d6 is a deuterium labeled Cariprazine. Cariprazine Cariprazine is an antipsychotic agent that exhibits high affinity for the D3 (Ki of 0.085 nM) and D2 (Ki of 0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (Ki of 2.6 nM)[1].

For research use only. We do not sell to patients.

Cariprazine-d<sub>6</sub> Chemical Structure

Cariprazine-d6 Chemical Structure

CAS No. : 1308278-67-2

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Based on 1 publication(s) in Google Scholar

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Description

Cariprazine-d6 is a deuterium labeled Cariprazine. Cariprazine Cariprazine is an antipsychotic agent that exhibits high affinity for the D3 (Ki of 0.085 nM) and D2 (Ki of 0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (Ki of 2.6 nM)[1].

IC50 & Target[1]

Dopamine D2 Receptor

0.49 nM (Ki)

Dopamine D3 Receptor

0.085 nM (Ki)

5-HT1A Receptor

2.6 nM (Ki)

Molecular Weight

433.45

Appearance

Solid

Formula

C21H26D6Cl2N4O
CAS No.
SMILES

O=C(N[[email protected]]1CC[[email protected]](CCN2CCN(C3=CC=CC(Cl)=C3Cl)CC2)CC1)N(C([2H])([2H])[2H])C([2H])([2H])[2H]
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Room temperature in continental US; may vary elsewhere.
Storage
Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
Purity & Documentation
References
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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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Keywords:

Cariprazine-d61308278-67-2RGH-188-d6Dopamine Receptor5-HT ReceptorSerotonin Receptor5-hydroxytryptamine ReceptorDeuteriumlabeledD2D35-HT1AInhibitorinhibitorinhibit

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