1. GPCR/G Protein
    Neuronal Signaling
  2. Dopamine Receptor
    5-HT Receptor
  3. Cariprazine D6

Cariprazine D6 (Synonyms: RGH-188 D6)

Cat. No.: HY-14763S
Handling Instructions

Cariprazine D6 (RGH-188 D6) is a deuterium labeled Cariprazine. Cariprazine Cariprazine is an antipsychotic agent that exhibits high affinity for the D3 (Ki of 0.085 nM) and D2 (Ki of 0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (Ki of 2.6 nM).

For research use only. We do not sell to patients.

Cariprazine D6 Chemical Structure

Cariprazine D6 Chemical Structure

Size Stock
100 mg   Get quote  
250 mg   Get quote  
500 mg   Get quote  

* Please select Quantity before adding items.

Top Publications Citing Use of Products
  • Biological Activity

  • Purity & Documentation

  • References

  • Customer Review

Description

Cariprazine D6 (RGH-188 D6) is a deuterium labeled Cariprazine. Cariprazine Cariprazine is an antipsychotic agent that exhibits high affinity for the D3 (Ki of 0.085 nM) and D2 (Ki of 0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (Ki of 2.6 nM)[1].

IC50 & Target[1]

Dopamine D2 Receptor

0.49 nM (Ki)

Dopamine D3 Receptor

0.085 nM (Ki)

5-HT1A Receptor

2.6 nM (Ki)

Molecular Weight

433.45

Formula

C₂₁H₂₆D₆Cl₂N₄O

SMILES

O=C(N[[email protected]]1CC[[email protected]](CCN2CCN(C3=CC=CC(Cl)=C3Cl)CC2)CC1)N(C([2H])([2H])[2H])C([2H])([2H])[2H]

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
  • No file chosen (Maximum size is: 1024 Kb)
  • If you have published this work, please enter the PubMed ID.
  • Your name will appear on the site.
  • Molarity Calculator

  • Dilution Calculator

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

Keywords:

Cariprazine D6RGH-188 D6Cariprazine D 6Cariprazine D-6Dopamine Receptor5-HT ReceptorSerotonin Receptor5-hydroxytryptamine ReceptorDeuteriumlabeledD2D35-HT1AInhibitorinhibitorinhibit

Your Recently Viewed Products:

Inquiry Online

Your information is safe with us. * Required Fields.

Product name

 

Salutation

Applicant name *

 

Email address *

Phone number *

 

Organization name *

Country or Region *

 

Requested quantity *

Remarks

Bulk Inquiry

Inquiry Information

Product name:
Cariprazine D6
Cat. No.:
HY-14763S
Quantity:
MCE Japan Authorized Agent: