1. Others GPCR/G Protein Neuronal Signaling
  2. Isotope-Labeled Compounds Dopamine Receptor 5-HT Receptor
  3. Cariprazine-d8

Cariprazine-d8  (Synonyms: RGH-188 d8)

Cat. No.: HY-14763S1 Purity: 99.51%
COA Handling Instructions

Cariprazine-d8 is a deuterium labeled Cariprazine. Cariprazine is a novel antipsychotic agent candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (Ki=2.6 nM).

For research use only. We do not sell to patients.

Cariprazine-d<sub>8</sub> Chemical Structure

Cariprazine-d8 Chemical Structure

CAS No. : 1308278-50-3

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1 mg USD 220 In-stock
5 mg USD 650 In-stock
10 mg USD 1050 In-stock
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Based on 1 publication(s) in Google Scholar

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Description

Cariprazine-d8 is a deuterium labeled Cariprazine. Cariprazine is a novel antipsychotic agent candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (Ki=2.6 nM).

IC50 & Target

D3 Receptor

 

Molecular Weight

435.46

Formula

C21H24D8Cl2N4O

CAS No.
Appearance

Solid

Color

White to off-white

SMILES

ClC1=C(C=CC=C1Cl)N2C([2H])([2H])C([2H])([2H])N(C([2H])([2H])C2([2H])[2H])CC[C@@H]3CC[C@H](CC3)NC(N(C)C)=O

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

4°C, sealed storage, away from moisture and light

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light)

Purity & Documentation
References
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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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Cariprazine-d8
Cat. No.:
HY-14763S1
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