1238697-26-1
1238697-26-1
Chemical Structure
Balipodect
Synonym(s): TAK-063
- CAS No.: 1238697-26-1
- Formula:C23H17FN6O2
- Molecular Weight:428.42
IUPAC Name: 1-(2-fluoro-4-(1H-pyrazol-1-yl)phenyl)-5-methoxy-3-(1-phenyl-1H-pyrazol-5-yl)pyridazin-4(1H)-one
InChIKey: KVHRYLNQDWXAGI-UHFFFAOYSA-N
SMILES: FC1=CC(N2N=CC=C2)=CC=C1N3N=C(C4=CC=NN4C5=CC=CC=C5)C(C(OC)=C3)=O
Biological Activity: Balipodect (TAK-063) is a selective, brain-penetrant and orally active PDE10A inhibitor with an IC50 of 0.30 nM. Balipodect shows >15000-fold selectivity over other PDEs. Balipodect elevates striatal cAMP and cGMP levels in mice. Balipodect can be used for the study of schizophrenia[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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Balipodect | 99.47% | Balipodect (TAK-063) is a selective, brain-penetrant and orally active PDE10A inhibitor with an IC50 of 0.30 nM. Balipodect shows >15000-fold selectivity over other PDEs. Balipodect elevates striatal cAMP and cGMP levels in mice. Balipodect can be used for the study of schizophrenia. | ||||||||||||||||||||
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Balipodect (Standard) | ≥98% | Balipodect (Standard) is the analytical standard of Balipodect. This product is intended for research and analytical applications. Balipodect (TAK-063) is a highly potent, selective and orally active PDE10A inhibitor with IC50 of 0.30 nM; >15000-fold selectivity over other PDEs. | ||||||||||||||||||||
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