130017-40-2
130017-40-2
Chemical Structure
K-756
- CAS No.: 130017-40-2
- Formula:C24H27N5O3
- Molecular Weight:433.50
IUPAC Name: 3-((1-(6,7-dimethoxyquinazolin-4-yl)piperidin-4-yl)methyl)-3,4-dihydroquinazolin-2(1H)-one
InChIKey: GWXCGEJJQFHPPA-UHFFFAOYSA-N
SMILES: O=C1NC2=C(C=CC=C2)CN1CC3CCN(C4=C5C=C(OC)C(OC)=CC5=NC=N4)CC3
Biological Activity: K-756 is a direct and selective tankyrase (TNKS) inhibitor, which inhibits the ADP-ribosylation activity of TNKS1 and TNKS2 with IC50s of 31 and 36 nM, respectively.
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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K-756 | 99.25% | K-756 is a direct and selective tankyrase (TNKS) inhibitor, which inhibits the ADP-ribosylation activity of TNKS1 and TNKS2 with IC50s of 31 and 36 nM, respectively. | ||||||||||||||||||||
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Keywords
