1356497-91-0
1356497-91-0
Chemical Structure
ST247
- CAS No.: 1356497-91-0
- Formula:C19H26N2O5S2
- Molecular Weight:426.55
IUPAC Name: methyl 3-(N-(4-(hexylamino)-2-methoxyphenyl)sulfamoyl)thiophene-2-carboxylate
InChIKey: MRWCGEOYGFZZCJ-UHFFFAOYSA-N
SMILES: O=C(C1=C(S(=O)(NC2=CC=C(NCCCCCC)C=C2OC)=O)C=CS1)OC
Biological Activity: ST247 a potent PPARβ/δ inverse agonist. ST247 has a higher affinity to PPARβ/δ. ST247 modulates expression of the activation marker CCL2 in the opposite direction. ST247 efficiently induces the interaction with corepressors. ST247 inhibits the agonist-induced transcriptional activity of PPARβ/δ[1].
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ST247 | 99.88% | ST247 a potent PPARβ/δ inverse agonist. ST247 has a higher affinity to PPARβ/δ. ST247 modulates expression of the activation marker CCL2 in the opposite direction. ST247 efficiently induces the interaction with corepressors. ST247 inhibits the agonist-induced transcriptional activity of PPARβ/δ. | ||||||||||||||||||||
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References
Keywords
