1627710-50-2
1627710-50-2
Chemical Structure
LJH685
- CAS. Nr.: 1627710-50-2
- Formula:C22H21F2N3O
- Molecular Weight:381.42
IUPAC Name: 2,6-difluoro-4-(4-(4-(4-methylpiperazin-1-yl)phenyl)pyridin-3-yl)phenol
InChIKey: IKUFKDGKRLMXEX-UHFFFAOYSA-N
SMILES: OC1=C(F)C=C(C2=C(C3=CC=C(N4CCN(C)CC4)C=C3)C=CN=C2)C=C1F
Biological Activity: LJH685 is a potent, ATP-competitive and selective RSK inhibitor, inhibits RSK1, 2, and 3 biochemical activities with IC50s of 6, 5, 4 nM, respectively[1].
| Art. -Nr. | Produktname | Reinheit | Beschreibung | Pricing | |||||||||||||||||||
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LJH685 | 99.64% | LJH685 is a potent, ATP-competitive and selective RSK inhibitor, inhibits RSK1, 2, and 3 biochemical activities with IC50s of 6, 5, 4 nM, respectively. | ||||||||||||||||||||
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Structural Analogs
-
Similarity Score 0.84
HY-19713LJI308 -
Similarity Score 0.62
HY-176941ALK2-IN-6 -
Similarity Score 0.59
HY-145045HPK1-IN-18 -
Similarity Score 0.58
HY-183720M4K2163 -
Similarity Score 0.57
HY-183005ActRIIB-IN-1 -
Similarity Score 0.57
HY-155939M4K2163 dihydrochloride -
Similarity Score 0.57
HY-183504ActRIIB-IN-3 -
Similarity Score 0.57
HY-151167LasR-IN-4 -
Similarity Score 0.57
HY-148234M4K2234 -
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