197894-84-1
197894-84-1
Chemical Structure
CI-1044
Synonym(s): PD-189659
- CAS No.: 197894-84-1
- Formula:C23H19N5O2
- Molecular Weight:397.43
IUPAC Name: (R)-N-(9-amino-4-oxo-1-phenyl-3,4,6,7-tetrahydro-[1,4]diazepino[6,7,1-hi]indol-3-yl)nicotinamide
InChIKey: XGXOSJSGDNPEEF-NRFANRHFSA-N
SMILES: O=C(C1=CC=CN=C1)N[C@H]2C(N3C4=C(CC3)C=C(N)C=C4C(C5=CC=CC=C5)=N2)=O
Biological Activity: CI-1044 is an orally active PDE4 inhibitor with IC50s of 0.29, 0.08, 0.56, 0.09 μM for PDE4A5, PDE4B2, PDE4C2 and PDE4D3, respectively.
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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CI-1044 | 98.02% | CI-1044 is an orally active PDE4 inhibitor with IC50s of 0.29, 0.08, 0.56, 0.09 μM for PDE4A5, PDE4B2, PDE4C2 and PDE4D3, respectively. | ||||||||||||||||||||
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Keywords
