2086257-77-2
2086257-77-2
Chemical Structure
VBIT-4
- CAS No.: 2086257-77-2
- Formula:C21H23ClF3N3O3
- Molecular Weight:457.87
IUPAC Name: N-(4-chlorophenyl)-4-hydroxy-3-(4-(4-(trifluoromethoxy)phenyl)piperazin-1-yl)butanamide
InChIKey: QYSQXVAEFPWMEM-UHFFFAOYSA-N
SMILES: O=C(NC1=CC=C(Cl)C=C1)CC(CO)N2CCN(C3=CC=C(OC(F)(F)F)C=C3)CC2
Biological Activity: VBIT-4 is an inhibitor of voltage-dependent anion channel 1 (VDAC1) oligomerization with a binding affinity (Kd) of 17 μM. VBIT-4, as an apoptosis inhibitor, can be used for therapeutic purposes in apoptosis-associated disorders, such as neurodegenerative and cardiovascular diseases[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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VBIT-4 | 99.86% | VBIT-4 is an inhibitor of voltage-dependent anion channel 1 (VDAC1) oligomerization with a binding affinity (Kd) of 17 μM. VBIT-4, as an apoptosis inhibitor, can be used for therapeutic purposes in apoptosis-associated disorders, such as neurodegenerative and cardiovascular diseases. | ||||||||||||||||||||
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VBIT-4 (Standard) | ≥98% | VBIT-4 (Standard) is the analytical standard of VBIT-4 (HY-129122). This product is intended for research and analytical applications. VBIT-4 is an inhibitor of voltage-dependent anion channel 1 (VDAC1) oligomerization with a binding affinity (Kd) of 17 μM. VBIT-4, as an apoptosis inhibitor, can be used for therapeutic purposes in apoptosis-associated disorders, such as neurodegenerative and cardiovascular diseases. | ||||||||||||||||||||
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