2104030-82-0
2104030-82-0
Chemical Structure
Brr2-IN-3
- CAS No.: 2104030-82-0
- Formula:C24H20N4O3S
- Molecular Weight:444.51
IUPAC Name: 6-benzyl-3-(3-(thiazol-5-ylmethoxy)phenyl)-4,6-dihydropyrido[4,3-d]pyrimidine-2,7(1H,3H)-dione
InChIKey: GAWVULNDIBAUHU-UHFFFAOYSA-N
SMILES: O=C1NC(C(CN1C2=CC=CC(OCC3=CN=CS3)=C2)=CN4CC5=CC=CC=C5)=CC4=O
Biological Activity: Brr2-IN-3 is a potent and selective Brr2 helicase allosteric Inhibitor. Brr2-IN-3 inhibits helicase activity in dose-dependent manner with an IC50 value of 1.3 μM[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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Brr2-IN-3 | 99.71% | Brr2-IN-3 is a potent and selective Brr2 helicase allosteric Inhibitor. Brr2-IN-3 inhibits helicase activity in dose-dependent manner with an IC50 value of 1.3 μM. | ||||||||||||||||||||
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Structural Analogs
-
Similarity Score 0.49
HY-112181KO-947 -
Similarity Score 0.47
HY-175232GL64 -
Similarity Score 0.47
HY-114116ML-109 -
Similarity Score 0.46
HY-18286NCGC00229600 -
Similarity Score 0.46
HY-176189CDK1-IN-7 -
Similarity Score 0.46
HY-148862Cavα2δ1&NET-IN-1 -
Similarity Score 0.45
HY-169054NCATS-SM4420 -
Similarity Score 0.45
HY-14440MP7 -
Similarity Score 0.45
HY-160617SIRT2-IN-14 -
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