2259641-46-6
2259641-46-6
Chemical Structure
DS-9300
- CAS No.: 2259641-46-6
- Formula:C25H26F3N5O3
- Molecular Weight:501.50
IUPAC Name: (2R,4R)-1-(4,4-difluoro-1-(4-methoxyphenyl)cyclohexane-1-carbonyl)-4-fluoro-N-(1H-pyrazolo[4,3-b]pyridin-5-yl)pyrrolidine-2-carboxamide
InChIKey: UCKDTCZSOLMOMQ-OXQOHEQNSA-N
SMILES: COC1=CC=C(C=C1)C2(CCC(F)(CC2)F)C(N3C[C@@H](C[C@@H]3C(NC4=NC5=C(NN=C5)C=C4)=O)F)=O
Biological Activity: DS-9300 is a potent, orally active, selective EP300/CBP HAT inhibitor with an IC50 value of 28 nM. DS-9300 has anticancer activity and can be used in prostate cancer disease research[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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DS-9300 | 99.83% | DS-9300 is a potent, orally active, selective EP300/CBP HAT inhibitor with an IC50 value of 28 nM. DS-9300 has anticancer activity and can be used in prostate cancer disease research. | ||||||||||||||||||||
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Structural Analogs
-
Similarity Score 0.91
HY-128875CBP/p300-IN-10 -
Similarity Score 0.86
HY-128367Ep300/CREBBP-IN-4 -
Similarity Score 0.77
HY-151812CBP/p300-IN-20 -
Similarity Score 0.77
HY-128362Ep300/CREBBP-IN-8 -
Similarity Score 0.76
HY-128364Ep300/CREBBP-IN-3 -
Similarity Score 0.76
HY-128363Ep300/CREBBP-IN-2 -
Similarity Score 0.69
HY-143442CBP/p300-IN-18 -
Similarity Score 0.60
HY-143441CBP/p300-IN-17 -
Similarity Score 0.58
HY-143443DS17701585 -
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