CBP/p300-IN-18
CBP/p300-IN-18 (compound 8) is a potent EP300/CBP HAT inhibitor with IC50s of 0.056, 0.46 µM for HAT EP300 and LK2 H3K27, respectively.
For research use only. We do not sell to patients.
- CAS No.: 2983027-64-9
- Formula: C25H27FN4O3
- Molecular Weight:450.51
-
Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
|
EP300 .056 μM (IC50) |
LK2 H3K27 0.46 μM (IC50) |
Chemical Information
-
CAS No. 2983027-64-9
-
Molecular Weight 450.51
-
Formula C25H27FN4O3
-
SMILES
O=C([C@@H]1N(C(C2(C3=CC=C(OC)C=C3)CCCC2)=O)C[C@H](F)C1)NC4=CC=CC5=C4C=NN5
-
Shipping
Room temperature in continental US; may vary elsewhere.
-
Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)