2361545-75-5
Chemical Structure
PKN3-IN-1
- CAS No.: 2361545-75-5
- Formula:C18H17IN2O3
- Molecular Weight:436.24
InChIKey: ZGFLIBPJHOZGNC-UHFFFAOYSA-N
SMILES: IC1=CC2=NC=CC(NC3=CC(OC)=C(C(OC)=C3)OC)=C2C=C1
Biological Activity: PKN3-IN-1 (compound 16) inhibits PKN3 (serine/threonine protein kinase 3) and GAK (cyclin G-associated kinase) with IC50 of 0.014 μM and Ki of 0.0044 μM respectively. PKN3-IN-1 is a potential tool compound to study the cell biology of PKN3 and its role in pancreatic and prostate cancer and T-cell acute lymphoblastic leukemia [1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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PKN3-IN-1 | 98.97% | PKN3-IN-1 (compound 16) inhibits PKN3 (serine/threonine protein kinase 3) and GAK (cyclin G-associated kinase) with IC50 of 0.014 μM and Ki of 0.0044 μM respectively. PKN3-IN-1 is a potential tool compound to study the cell biology of PKN3 and its role in pancreatic and prostate cancer and T-cell acute lymphoblastic leukemia . | ||||||||||||||||||||
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