3572-80-3
Chemical Structure
Cyclazocine
- CAS No.: 3572-80-3
- Formula:C18H25NO
- Molecular Weight:271.40
IUPAC Name: 3-(cyclopropylmethyl)-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2,6-methanobenzo[d]azocin-8-ol
InChIKey: YQYVFVRQLZMJKJ-UHFFFAOYSA-N
SMILES: OC1=CC=C2C(C3(CCN(C(C3C)C2)CC4CC4)C)=C1
Biological Activity: Cyclazocine is a μ, δ, and κ opioid receptor modulator with Ki values of 0.32, 1.1, and 0.18 nM, respectively. Cyclazocine exhibits "mixed" pharmacological activities, acting as a μ-partial antagonist, κ-agonist, and low-affinity δ ligand. Cyclazocine shows antinociceptive activity in mice. Cyclazocine can be used in studies on psychoactive substance addiction[1].
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Cyclazocine | Cyclazocine is a μ, δ, and κ opioid receptor modulator with Ki values of 0.32, 1.1, and 0.18 nM, respectively. Cyclazocine exhibits "mixed" pharmacological activities, acting as a μ-partial antagonist, κ-agonist, and low-affinity δ ligand. Cyclazocine shows antinociceptive activity in mice. Cyclazocine can be used in studies on psychoactive substance addiction. | |||||||||||||||||||||
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Keywords
