1. Epigenetics
  2. Epigenetic Reader Domain
  3. CBP/P300 bromodomain inhibitor-3

CBP/P300 bromodomain inhibitor-3 

Cat. No.: HY-136920
Handling Instructions

CBP/P300 bromodomain inhibitor-3 is a potent inhibitor of the CBP/P300 family of bromodomains. CBP/P300 bromodomain inhibitor-3 inhibits CBP (IC50=0.01-0.1 µΜ) and BRD4 (IC50=1-1000 µΜ) activity.

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CBP/P300 bromodomain inhibitor-3 Chemical Structure

CBP/P300 bromodomain inhibitor-3 Chemical Structure

CAS No. : 2304416-91-7

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Description

CBP/P300 bromodomain inhibitor-3 is a potent inhibitor of the CBP/P300 family of bromodomains. CBP/P300 bromodomain inhibitor-3 inhibits CBP (IC50=0.01-0.1 µΜ) and BRD4 (IC50=1-1000 µΜ) activity[1].

IC50 & Target[1]

CBP

0.01-0.1 μM (IC50)

BRD4

1-1000 μM (IC50)

Molecular Weight

461.55

Formula

C₂₇H₃₁N₃O₄

CAS No.

2304416-91-7

SMILES

O=C(N1[[email protected]@H](C)CCC2=C1C=CC3=C2N=C(CC4=CC=CC=C4)N3[[email protected]@H]5C[[email protected]@H](C(O)=O)CCC5)OC

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Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Keywords:

CBP/P300 bromodomain inhibitor-3Epigenetic Reader DomainInhibitorinhibitorinhibit

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CBP/P300 bromodomain inhibitor-3
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HY-136920
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