1. Epigenetics
  2. Histone Acetyltransferase
  3. CBP/p300-IN-16

CBP/p300-IN-16 

Cat. No.: HY-143440
Handling Instructions

CBP/p300-IN-16 (compound 1) is a potent EP300/CBP HAT inhibitor with IC50s of 0.61, 2.24 µM for HAT EP300 and LK2 H3K27, respectively.

For research use only. We do not sell to patients.

CBP/p300-IN-16 Chemical Structure

CBP/p300-IN-16 Chemical Structure

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Description

CBP/p300-IN-16 (compound 1) is a potent EP300/CBP HAT inhibitor with IC50s of 0.61, 2.24 µM for HAT EP300 and LK2 H3K27, respectively[1].

IC50 & Target[1]

EP300

0.61 μM (IC50)

LK2 H3K27

2.24 μM (IC50)

Molecular Weight

449.54

Formula

C26H31N3O4

SMILES

O=C(N1CCOC[[email protected]](CC2=CC=CC3=C2C=NN3)C1)C4(C5=CC=C(OC)C=C5)CCOCC4

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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The dilution calculator equation

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This equation is commonly abbreviated as: C1V1 = C2V2

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Product Name:
CBP/p300-IN-16
Cat. No.:
HY-143440
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