CP-464709
CP-464709 is a Ghrelin receptor agonist that can penetrate the blood-brain barrier. CP-464709 causes an increase in blood pressure by activating pre sympathetic neurons in the spinal cord. CP-464709 causes biphasic blood pressure response when administered intravenously, while intrathecal administration only causes pressor. CP-464709 can be used for research on cardiovascular conditions.
Nur für Forschungszwecke. Wir verkaufen nicht an Patienten.
- CAS. Nr.: 193272-70-7
- Formel: C28H31F5N6O4
- Molecular Weight:610.58
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Speicherung:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biologische Aktivität
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Chemical Information
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Help & FAQs
Biologische Aktivität
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| Pituitary gland cell | EC50 |
3 nM
Compound: 4, (CP-464709-18)
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In vitro effective concentration required for 50% stimulation of GH release in rat pituitary cell cultures.
In vitro effective concentration required for 50% stimulation of GH release in rat pituitary cell cultures.
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[PMID: 12392732] |
Chemical Information
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CAS. Nr. 193272-70-7
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Molecular Weight 610.58
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Formel C28H31F5N6O4
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SMILES
CC(C)(N)C(N[C@H](COCC1=CC=C(F)C=C1F)C(N(C[C@]23CC4=NC=CC=C4)CCC2=NN(CC(F)(F)F)C3=O)=O)=O
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Versand
Room temperature in continental US; may vary elsewhere.
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Speicherung
Please store the product under the recommended conditions in the Certificate of Analysis.
Reinheit & Dokumentation
Verweise
Calculators
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)
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