BMS-986034
BMS-986034 is an orally active ingredient (API) that is an agonist of GPR119..
Nos produits utilisent uniquement pour la recherche. Nous ne vendons pas aux patients.
- CAS No.: 1492631-88-5
- Formule: C24H24Cl2N6O4
- Masse moléculaire:531.39
-
Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Activité biologique
GPR119[1]
|
Cell Line
|
Type | Value | Description | References |
|---|---|---|---|---|
| HEK293 | EC50 |
3 nM
Compound: 4
|
Agonist activity at human-mouse chimeric GPR119 expressed in tetracycline-induced Flp-In-T-Rex-HEK293 cells assessed as accumulation of cAMP after 50 mins by HTRF assay
Agonist activity at human-mouse chimeric GPR119 expressed in tetracycline-induced Flp-In-T-Rex-HEK293 cells assessed as accumulation of cAMP after 50 mins by HTRF assay
|
[PMID: 24900860] |
Chemical Information
-
CAS No. 1492631-88-5
-
Masse moléculaire 531.39
-
Formule C24H24Cl2N6O4
-
SMILES
O=C1C=C(C(Cl)=CN1C2=NC(C)=C(C=C2)N3C([C@@H](CC3)O)=O)OC4CCN(CC4)C5=NC=C(C=N5)Cl
-
Livraison
Room temperature in continental US; may vary elsewhere.
-
Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)