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Cat. No.: HY-125055A

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CD08108

CD08108 is a selective MC1R full agonist with an EC₅₀ of 70 nM against hMC1R. CD08108 participates in the melanogenesis process. CD08108 promotes cell proliferation. CD08108 can be used in studies related to vitiligo, subcutaneous diseases and photosensitive diseases.

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CAS No.: 1417342-67-6
Formule: C₃₁H₃₈N₄O₄
Masse moléculaire:530.67

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Please store the product under the recommended conditions in the Certificate of Analysis.

CD08108 Chemical Structure

CAS No.: 1417342-67-6

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Use of MCE Products

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Activité biologique
- Description
- IC₅₀ & Target
- In Vitro
Chemical Information
Pureté et documentation
Références
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Description

IC₅₀ & Target

^[2]

MC1R

70 nM (EC₅₀)

MC4R

4500 nM (EC₅₀)

Voir tous les produits spécifiques à Isoform Melanocortin Receptor :

In Vitro

CD08108 acts as a selective hMC1R agonist with an EC₅₀ of 70 nM, showing 64-fold higher potency for hMC1R compared to hMC4R^[2].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Related Protocols :

Chemical Information

CAS No. 1417342-67-6
Masse moléculaire 530.67
Formule C₃₁H₃₈N₄O₄
SMILES

O(CC1CC1)C2(CN(C([C@@H](CC3=CC=C(OC)C=C3)NC(CCC=4NC=NC4C)=O)=O)C2)C5=C(C)C=CC=C5
Livraison

Room temperature in continental US; may vary elsewhere.
Stockage

Please store the product under the recommended conditions in the Certificate of Analysis.

Pureté et documentation

Instruction de manipulation (2659 KB)

Références

[1]. Boiteau J G, et al. Development of a Kilogram-Scale Synthesis of a Novel MC1R Agonist[J]. Organic Process Research & Development, 2015, 19(6): 646-651.

[2]. Mun Y, et al. Melanocortin 1 Receptor (MC1R): Pharmacological and Therapeutic Aspects. Int J Mol Sci. 2023;24(15):12152. Published 2023 Jul 29. [Content Brief]

[3]. Mun Y W, et al. Melanocortin 1 Receptor (MC1R): Potentials as therapeutic targets[J]. 2023.

Calculators

Calculateur de molarité

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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Calculateur de dilution

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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100 mg

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- In Vitro
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CD08108

Voir tous les produits spécifiques à Isoform Melanocortin Receptor

Activité biologique

Description

IC50 & Target

In Vitro

Chemical Information

Pureté et documentation

Références

Calculators

Help & FAQs

CD08108 Related Classifications

HY-125055A Related Classifications

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