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Cat. No.: HY-10051

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GR203040

Name: GR203040
Brand: MedChemExpress
SKU: HY-10051
Price: 370.00 USD
Availability: InStock
Rating: 5 (1 reviews)

GR203040 is an orally active NK₁ receptor antagonist with a pK_i of 10.3. GR203040 shows potent antiemetic activity.

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CAS No.: 168398-02-5
Formule: C₂₀H₂₆Cl₂N₆O
Masse moléculaire:437.37

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Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (271 KB)

GR203040 Chemical Structure

CAS No.: 168398-02-5

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Activité biologique
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Chemical Information
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Description

GR203040 is an orally active NK₁ receptor antagonist with a pK_i of 10.3. GR203040 shows potent antiemetic activity^[1].

IC₅₀ & Target

pKi: 10.3 (NK₁ receptor)^[1]

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Chemical Information

CAS No. 168398-02-5
Masse moléculaire 437.37
Formule C₂₀H₂₆Cl₂N₆O
SMILES

COC1=CC=C(N2N=NN=C2)C=C1CN[C@@H]3[C@H](C4=CC=CC=C4)NCCC3.[H]Cl.[H]Cl
Livraison

Room temperature in continental US; may vary elsewhere.
Stockage

Please store the product under the recommended conditions in the Certificate of Analysis.

Pureté et documentation

Select Batch:

Pureté: 99.98%

Assay: 99.98%

ee.: 99.98%

Fiche technique (271 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Instruction de manipulation (2659 KB)

Références

[1]. Ward P, et al. Discovery of an orally bioavailable NK1 receptor antagonist, (2S,3S)-(2-methoxy-5-tetrazol-1-ylbenzyl)(2-phenylpiperidin-3-yl)amine (GR203040), with potent antiemetic activity. J Med Chem. 1995 Dec 22;38(26):4985-92. [Content Brief]

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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100 mg

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GR203040

Voir tous les produits spécifiques à Isoform Neurokinin Receptor

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